• General • Film-coating materials polymers, additives, formulation—including solutions and suspension properties • Physicochemical properties of coating systems including interactions o
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16 Bibliography Michael E.Aulton
A PHARMACEUTICAL FILM COATING PUBLICATIONS BIBLIOGRAPHY
This chapter contains a comprehensive listing of research papers, reviews, book chapters and theses covering the subject of pharmaceutical film coating Coating is a very extensive subject and so this bibliography is restricted to those publications of direct pharmaceutical relevance or authorship Non-pharmaceutical polymer science or coating processes of other industries are not included
While the listing is extensive, it is by no means exhaustive Indeed, the author would welcome
notification of any missing articles in order that this work can be included in the next edition Similarly, notification of any errors in these listings would be welcomed
For convenience, the published work is categorized into the following subjects; some papers fall into more than one category
• General
• Film-coating materials (polymers, additives, formulation—including solutions and suspension properties)
• Physicochemical properties of coating systems (including interactions of polymers and additives, and thermomechanical properties)
• Coating processes
• Wetting and adhesion
• Mechanical properties
• Quality of coats (including defects, gloss, surface roughness and colour)
• Permeability (to gases and water vapour)
• Drug release characteristics
• Stability
• Miscellaneous pharmaceutical coating publications: Bioadhesion; Coating of hard gelatin
capsules
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General
Banker, G.S (1966) Film coating theory and practice J Pharm Sci 55(1), 81–89
Banker, G.S., Peck, G., Jan, S., Pirakitikulr, P & Taylor, D (1981) Evaluation of hydroxypropyl
cellulose and hydroxypropyl methyl cellulose as aqueous based film coatings Drug Dev Ind Pharm.
7(6), 693–716
Ellis, J.R., Prillig, E.B & Endicott, C.J (1970) Tablet coating In Lachman, L (ed.), The theory and
practice of industrial pharmacy, Lea and Fabinger, Philadelphia, PA, USA, cha p 10 , 197–225
Hogan, J.E (1978) Aqueous cellulosic film coating of tablets J Pharm Pharmacol 30 Suppl., 88P
Hogan, J.E (1988) Tablet coating In Pharmaceutics: the science of dosage form design (ed Aulton,
M.E.), Churchill-Livingstone, Edinburgh
McGinity, J.W (ed.) (1989) Aqueous polymeric coatings for pharmaceutical dosage forms, Marcel
Dekker, New York, 424pp
Onions, A (1986) Films from water-based colloidal dispersions Manuf Chem 57(3), 55–59
Onions, A (1986) Films from water-based colloidal dispersions Manuf Chem 57(4), 66–67
Pickard, J.F & Rees, J.E (1972) Modern trends in pharmaceutical coating Pharm Ind 34(11), 833–
839
Pickard, J.F & Rees, J.E (1974) Film coating: 1 Formulation and process considerations in film
coating Manuf Chem 54(4), 19–22
Porter, S.C (1978) Aqueous film coating: an overview Pharm Technol 3(9), 55–59
Porter, S.C (1981) Tablet coating I Drug Cosmet Ind 129(5), 46–53, 86–93
Porter, S.C (1981) Tablet coating II Drug Cosmet Ind 129.
Porter, S.C (1981) Tablet coating III Drug Cosmet Ind 129(8), 40–44, 87–88
Porter, S.C (1981) Tablet coating IV Drug Cosmet Ind 129(9), 50–58
Porter, S.C & Hogan, J.E (1984) Tablet film-coating Pharm Int 5(5), 122–127
Tondachi, M., Hoshi, N & Sekigawa, F (1977) Tablet coating in an aqueous system Drug Dev Ind
Pharm 3(3), 227–240
Film coating materials (polymers, additives, formulation—including solutions and
suspension properties)
Banker, G.S & Peck, G.E (1981) The new, water-based colloidal dispersions Pharm Technol 5(4).
Banker, G.S., Peck, G.E., Jan, S., Pirakitikulr, P & Taylor, D (1981) Evaluation of hydroxypropyl
cellulose and hydroxypropyl methyl cellulose as aqueous based film coatings Drug Dev Ind Pharm.
7(6), 693–716
Banker, G.S., Peck, G.E., Williams, E., Taylor, D & Pirakitikulr, P (1982) Microbiological
considerations of polymer solutions used in aqueous film coating Drug Dev Ind Pharm 8(1), 41–
51
Benita, S (1987) Cellulose hydrogen phthalate A coating polymer in controlled release dosage forms
Pharm Acta Helv 62, 255–261
Bergisadi, N (1986) Two new derivatives of alginic acid for tablet coating S.T.P Pharma 2(18), 620–
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Bindschaedler, C, Gurny, R & Doelker, E (1983) Notions theoriques sur la formation des films obtenus
a partir de microdispersions aqueuses et application a l’enrobage Labo-Pharma Probl Tech 31(331),
389–394
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aqueous latexes Pharm Res 6(8), 725–730
Chang, R.-K (1990) Preparation and evaluation of shellac pseudolatex as an aqueous enteric coating
system for pellets Int J Pharmaceut 60, 171–173
Chang, R.-K (1990) A comparison of rheological and enteric properties among organic solutions,
ammonium salt aqueous solutions and latex systems Pharm Technol 14(10), 62–70
Chopra, S.K & Tawashi, R (1982) Tack behavior of coating solutions I J Pharm Sci., 71(8), 907–
911
Chopra, S.K & Tawashi, R (1984) Tack behavior of coating solutions II J Pharm Sci 73(4), 477–
481
Chopra, S.K & Tawashi, R (1985) Tack behavior of coating solutions III J Pharm Sci 74(7), 746–
749
Delonca, H (1989) Etude de films à base d’hydroxypropylméthylcellulose phtalate (HP55) I: Films
isolés J Pharm Belg 44, 17–35
Delonca, H (1989) Etude de films à base d’hydroxypropylméthylcellulose phtalate (HP55) II: Films
appliqués J Pharm Belg 44, 101–108
Eskilsson, C., Appelgren, C & Bogentoft, C (1976) A note on the properties of
ethylcellulose-propylene glycol membranes Acta Pharm Suec 13, 285–288
Gumowski, F., Doelker, E & Gurny, R (1987) The use of a new redispersible aqueous enteric coating
material Pharm Technol 11, 26–32
Hogan, J.E (1983) Additive effects on aqueous film coatings Manuf Chem 54(4), 43–47
Joachim, J (1990) Etudes comparative de deux filmogènes: acétophtalate de cellulose et l’Aquatéric
Pharm Acta Helv 65, 311–314
Kanig, J.L & Goodman, H (1962) Evaluative procedures for film-forming materials used in
pharmaceutical applications J Pharm Sci 51, 77–82
Kent, D.J & Rowe, R.C (1978) Solubility studies on ethyl cellulose used in film coating J Pharm
Pharmacol 30, 808–810
Kovács, B & Merényi, G (1990) Evaluation of tack behaviour of coating solutions Drug Dev Ind
Pharm 16(15), 2303–2323
Kumar, V & Banker, G.S (1993) Chemically-modified cellulosic polymers Drug Dev Ind Pharm 19
(1 and 2), 1–31
Lehmann, K (1986) Mischbarkheit wässriger Poly(meth)acrylat-Dispersionen für
Arzneimittelüberzüge Pharm Ind 48, 1182–1183
Lehmann, K (1989) Chemistry and application properties of polymethacrylate coating systems In
McGinity, J.W (ed.), Aqueous polymeric coatings for pharmaceutical dosage forms, Marcel Dekker,
New York, 153–245
Trang 5Lejeune, B (1987) Emploi du rouge de betterave pour la coloration de comprimés pelliculés S.T.P
Pharma 3, 400–406
Lindholm, T (1982) Controlled release tablets Part 3: Ethylcellulose coats containing surfactant and
powdered matter Pharm Ind 44, 937–941
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Lindholm, T., Huhtikangas, A & Saarikivi, P (1984) Organic solvent residues in free ethyl cellulose
films Int J Pharmaceut 21, 119–121
Munden, B.J., DeKay, H.G & Banker, G.S (1964) Evaluation of polymeric materials I: Screening of
selected polymers as film coating agents J Pharm Sci 53, 395–401
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copolymers J Pharm Pharmacol 43, 198–200
Opota, O (1988) Comportement rhéologique des solutions aqueuses d’hydroxypropylcellulose
Influence de la concentration et de la masse moléculaire Pharm Acta Helv 63, 26–32
Osterwald, H.P (1982) Wirkungsweise und Optimierungsmöglichkeiten der Anwendung von
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Pharm Acta Helv 63(2), 46–53
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enteric coating properties S.T.P Pharma Sci 1, 267–271
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Technol 4(3), 66–75
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50(10), 1245–1249
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Rosoff, M & Sheen, P.C (1983) Abrasion and polymorphism of titanium dioxide in coating
suspensions J Pharm Sci 72(12), 1485
Rowe, R.C (1980) The molecular weight and molecular weight distribution of hydroxypropyl
methylcellulose used in film coating of tablets J Pharm Pharmacol 32, 116–119
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19, 157–160
Rowe, R.C (1982) Molecular weight studies on hydroxypropyl methylcellulose phthalate (HP55) Acta
Pharm Technol 28(2), 127–130
Rowe, R.C (1982) Some fundamental properties of polymeric materials and their application in film
coating formulations—a review Int J Pharm Tech Prod Mfr 3(1), 3–8
Rowe, R.C (1983) The orientation and alignment of particles in tablet film coatings J Pharm
Pharmacol 35, 43–44
Rowe, R.C (1984) Materials used in the film coating of oral dosage forms In Florence , A.T (ed.),
Materials used in pharmaceutical formulation Critical Reports in Applied Chemistry 6, 1–36
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Rowe, R.C (1988) Characterisation of the structure of filled polymer film coating using ion beam
etching Int J Pharmaceut 47, 205–208
Rowe, R.C (1992) Molecular weight dependence of the properties of ethyl cellulose and hydroxypropyl
methylcellulose films Int J Pharmaceut 88, 405–408
Rowe, R.C & Forse, S.F (1983) The refractive indices of polymer film formers, pigments and additives
used in tablet film coating: their significance and practical application J Pharm Pharmacol 35,
205–207
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55, 157–160
Tardieu, M (1992) Etude comparative de dispersions aqueuses de polymerès gastrorésistants
entérosolubles Pharm Acta Helv 67, 29–32
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lacquer film coating Drug Dev Ind Pharm 15(2), 165–185
Utsumi, I., Ida, T., Takahashi, S & Sugimoto, N (1961) Studies on protective coatings IX:
polyvinylpyridine derivatives J Pharm Sci 50, 592–597
Venkateswarlu, V., Kokate, C.K., Rambhau, D & Veeresham, C (1993) Pharmaceutical investigations
of a film forming material isolated from roots of salacia macrosperma Drug Dev Ind Pharm 19(4),
461–472
Wan, L.S.C (1991) A simple method to assess the tack of coating formulations S.T.P Pharma 2, 174–
180
Wan, L.S.C (1991) An application of tack measurement to fluidized bed coating S.T.P Pharma 2,
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Gibson, S.H.M., Rowe, R.C & White, E.F.T (1988) Characterisation of the structure of filled polymer
film coatings using ion beam etching Int J Pharmaceut 47, 205–208
Gibson, S.H.M., Rowe, R.C & White, E.F.T (1988) Quantitative assessment of additive-polymer interaction in pigmented hydroxypropyl methylcellulose formulations using immersion calorimetry
Int J Pharmaceut 48, 113–117
Humeke-Bogner, R., Liu, J.-C & Chien, Y.W (1988) Methods for determining partial solubility
parameters of potential film-coating polymers Int J Pharmaceut 42, 199–209
Jacobsson, S & Hagman, A (1990) Characterization of polymers used as pharmaceutical excipients by
dynamic headspace gas chromatography-mass spectrometry Drug Dev Ind Pharm 16(17), 2547–
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dynamic mechanical analysis J Pharm Sci 79, 845–848
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Lafferty, S.V., Summers, M.P., Mackey, R & Newton, J.M (1990) The application of dynamic
mechanical thermal analysis to study the physical properties of free polymeric films J Pharm
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analysis I Penetration mode Int J Pharmaceut 20, 295–305
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