... activity andinverse agonism in a family C G -protein- coupled receptor. J. Biol.Chem. 275, 29547–29555.52. Chen, R., Mukhin, Y. V., Garnovskaya, M.N., Thielen, T.E.,Iijima, Y. , Huang, C., Raymond, ... Department of Medicinal Chemistry, The Royal Danish School of Pharmacy,Copenhagen, Denmark;2Laboratory of Molecular Cardiology, Copenhagen University Hospital, University of Copenhagen,Copenhagen, ... receptors.Neuropharmacology 38, 1431–1476.4. Brown, E.M. (1999) Physiology and pathophysiology of theextracellular calcium-sensing receptor. Am.J.Med.106, 238–253.5. Mo¨hler, H. & Fritschy, J M. (1999)...