Pharmaceutical Substances Syntheses, Patents, Applications - Part 13 potx
Pharmaceutical Substances Syntheses, Patents, Applications - Part 2 potx
... levulinoyloxyacetate
benzyl 1 2- ( 4-methoxyphenylhydrozano )-
'=?'
benzyl
(5-meVloxy -2 - methyl-3-lndolyl-
4-chloro-
benzoyl chloride
benzyl
[I
-( 4-chlorobenzoyl )-5 -methoxy-
2- methyl-3-indolylocetoxy]acetate ... C,yH22N20S MW: 326 .46 EINECS: 23 6-6 6 1-9
LD,,: 517 mgkg (M, p.0.)
CN:
1-[ l 0-[ 2- ( dimethylamino)propyl ]-1 0H-phenothiazin -2...
Pharmaceutical Substances Syntheses, Patents, Applications - Part 8 potx
... 5 58 8- 1 6-9 MF: C,,H14C1N304S3
MW:
383 .90 EINECS: 22 6-9 9 4 -8
CN:
6-chloro-3,4-dihydro- 3-[ (2-propenylthio)methy1 ]-2 H-
1,2,4-benzothiadiazine-7-sulfonamide
1,
l-dioxide
6-amino-4-chloro- chloroocetaldehyde ... hydrochloride
CH3-CO-NH-NH2
,
butanol
-
acetohydrazide
2-0 x 0-2 .3-dihydro-lH-
2-thioxo-2,3-dihydro- 7-chloro-5-phenyl-3H-
1.4-benzodiazepin...
Pharmaceutical Substances Syntheses, Patents, Applications - Part 13 potx
...
1-cyclohexyl-3-morpholinyl-
ethyl-corbodiimide
+
N
b
VII
H-Val-Tyr-Val-His-Pro-Phe-0-CH
(VI)
I-N
ti2,
~d-C.CH~OH
-m
H H
Z-Asn-Arg(N02)-Val-Tyr-Val-His-Pro-Phe-0-CH
(W)
130
A
Apalcillin ...
Z-N
0
111
+
HN,COOH
\INYN/~0,
H
H
Z
-Asn-Arg(N0,)-OH
(N)
DMF,
1
-cyclahexyl- 3-
morpholinylethyl-carbodiimide
+
I1
v
Z-Val-Tyr-Val-His-Pro-Phe-0-CH
(V)
DMF,
1-cyc...
Pharmaceutical Substances Syntheses, Patents, Applications - Part 22 potx
...
1,2,3.4-tetrahydro-6,7-dimethoxy-
2-isoquinolineprapionote
[Ill)
ethyl 1.3.4.6.7.1 1 b-hexohydm-
N.N-diethyl-1.3.4.6.7,ll
b-hexahydro-9.10.
dimethoxy- 2-0 x 0-2 H-
9,lO-dimethaxy- 2-0 x 0-2 H-
benzo[o]quinalizine- ...
6-chloro- 3-[ [(phenylmethyl)thio]methyl ]-2 H-1,2,4-benzothiadiazine-7-sulfonamide
1,l-dioxide
5-chloro-2.4-diomino- chloro-
7-ominonulfonyl-6-chloro-...
Pharmaceutical Substances Syntheses, Patents, Applications - Part 25 potx
...
RN:
3463 3-3 4-6 MF: C,,H,,F,O, MW: 292.33
CN:
(R*,S* )-4 ,4&apos ;-( 1-ethyl-2-methyl-l,2-ethanediyl)bis[2-fluorophenol]
3-chloro- 2-
trans-2.3-bis(3-fluora-4-methoxy-
pentanone phenyl )-2 -pentene ... 20 0-3 9 9-3
CN:
[3aS-(3aa,4~,6aa)]-hexahydro-2-oxo-1H-thieno[3,4-d]imidazole-4-pentanoic
acid
fumoric ocid mesa-2.3-dibromo- cis-1,3-dibenzyl-
succinic ocid 2-axo...
Pharmaceutical Substances Syntheses, Patents, Applications - Part 27 potx
... ocetate. O°C
XI1
-
XI11
3-( brornoocetyl )-
5-chloro- 2-
thiophenesulfonomide
(XlIl)
K2C03, DMSO
XN
+
X
b
4-hydroxy- 2-( 3-rnethoxy-
propy1 )-2 H- thieno[3.2-el-
1,2-thiozine 1.1-dioxide (XV) ... oxolate
Z-picaline 2-picoline ethyl 2-pyridyl-
1
-axide pyruvate 1'-oxide
(In)
4-brornophenyl-
hydrozine hydrochloride
ethyl 5-brorno- 3-
(2-pyridy1)ind...
Pharmaceutical Substances Syntheses, Patents, Applications - Part 42 potx
... 143 1 .O6
CN:
N-Acetyl- 3-( 2-naphthalenyl )-~ -alanyl-4-choro-~-phenyaanyl- 3-( 3-pyridinyl )-~ -alanyl-~-seryl- ~-
tyrosyl- ~-( aminocarbonyl )-~ -ornithyl-~-leucyl-~-arginy ~-~ -prolyl-~-alaninamide
... 1765 0-9 8-5 MF:
C5RH73N1302LS2
MW: 1352 .42
LD,,:
1012 mgkg
(M,
i.v.)
CN:
5-oxo-~-prolyl-~-glutaminyl-~-a-asparty-O-sulfo-~-tyrosyl-~-threonylglycyl-~-tr...
Pharmaceutical Substances Syntheses, Patents, Applications - Part 46 potx
... bronchodilator
RN: 449 9-4 0-5 MF: C7H7N402. C5H,,N0 MW: 283.33 EINECS: 22 4-7 9 8-7
CN:
2-hydroxy-N,N,N-trimethylethanaminium,
salt with
3,7-dihydro-l,3-dimethyl-IH-purine-2,6-dione
(1:l)
a-Chymotrypsin ...
CN:
(2R-trans )-2 -( 3,4-dihydroxyphenyl )-3 ,4-dihydro-2H-I-benzopyran-3,5,7-triol
Cholestyramine
C
453
Formulation(s):
tabl. 250 mg, 500 mg
Trade Name(s):
D...
Pharmaceutical Substances Syntheses, Patents, Applications - Part 47 potx
... 5986 5-1 3-3 MF: C,,Hll,N,,O,, MW: 1202.64
CN:
[R-[R*,S *-( E)]]-cyclic(~-alanyl-~-alanyl-N-methyl-~-leucyl-N-methyl-~-leucyl-N-methyl-~-valyl- 3-
hydroxy-N,4-dimethyl- ~-2 -amino-6-octenoyl-~-a-aminobutyryl-N-methylglycyl-N-methyl-~-leucyl- ~- ...
hydrochloride
methyl 5-cyclohexyl-
3-methyl- 5-0 x 0-2 -
pentenoote (mixture
with
the 3-pentenoote:
from methyl 4-me...
Pharmaceutical Substances Syntheses, Patents, Applications - Part 56 potx
...
l 0-[ 3-( dimethylamino )-2 -methylpropyl ]-1 0H-phenothiazine-2-carbonitrile
Z-chloropheno-
thiozine
P-cyanopheno-
thiozine
1.
NaNH2, xylene
2.
cl&i:3
CH3
I
2.
1
-chloro-3-dimethyl-
amino-2-methyl-
Cyamemazine ... tonic
RN: 63 3-4 7-6 MF: C,3H24N202
MW:
240.35 EINECS: 2
1
1-1 9 3-8
CN:
N-[ 1-[ (dirnethylamino)carbonyI]propyl]-N-propyl-2-butenamid...
Pharmaceutical Substances Syntheses, Patents, Applications - Part 73 potx
...
-dimethylethyl)phenyl ]-4 -[ 4-( diphenylmethoxy)
1 -piperidinyl ]- 1-butanone
4-tert-butyl-w-chloro- 4-hydroxypiperidine
1
-[ 3-( 4-tert-butylbenzoyl )-
butyrophenone
(I)
propyll-4-hydroxypiperidine
-( [I)
3.
1
______, ...
1-[ 1-[ 4-( 4-fluorophenyl )-4 -oxobutyl ]-1 ,2,3,6-tetrahydro-4-pyridinyl ]-1 ,3-dihydro-2H-ben~imidazo 1-2 -one
ethyl
1
-...
Pharmaceutical Substances Syntheses, Patents, Applications - Part 78 potx
... 2997 5-1 6-4 MF:
C,,Hl1ClN4 MW: 294.75 EINECS: 24 9-9 8 2-4
LD,,,: 600 mglkg (M, p.0.);
2500 mglkg (R, p.0.)
CN:
8-chloro-6-phenyl-4H-[1,2,4]tnazolo[4,3-a][l,4]benzodiazepine
2-omino-5-chloro- ...
methyl 3-( 4-hydroxy- epichloro-
pheny1)propionote hydrin
methyl
3-[ 4-( 2.3-epoxy-
propoxy)phenyl]propionate
(I)
778
E
Estazolam
Reference(s):
EP 41 491 (Hassle; a...
Pharmaceutical Substances Syntheses, Patents, Applications - Part 79 potx
... estrogen
RN: 5 3-1 6-7
MF:
Cl,HzzOz
MW:
270.37 EINECS: 20 0-1 6 4-5
CN:
3-hydroxyestra-1,3,5(10)-trien-17-one
oxide
androatenolone
3.17-dioxo-1. 4-
ondrostadiene
(n)
$17-dioxo-1.4. 6-
ondrostatnene ... 9 0-5 4-0 - MF: C2,H2,N02 MW: 325.45 EINECS: 20 2-0 0 2-9
CN:
l-[ 2-[ 2-( diethylamino)ethoxy]phenyl ]-3 -phenyl-l-propanone
hydrochloride
RN: 21...
Pharmaceutical Substances Syntheses, Patents, Applications - Part 87 potx
...
6,8-Difluoro-l-(2-fluoroethyl)-l,4-dihydro- 7-( 4-rnethyl-1-piperazinyl )-4 -oxo-3-quinolinecarboxylicacid
monohydrochloride
RN: 7966 0-5 3-0 MF: C,,H,,F,N,O,
.
HCl MW: 405.80
6,7,8-trifluoro- 4- ...
(6R-ci.~ )-7 -[ [[(difluoromethyl)thio]acetyl]amino ]-3 -[ [[l-(2-hydroxyethyl)-lH-tetrazol-5-yl]thio]methyl ]-
7-methoxy-8-oxo-5-oxa-1-azabicyclo[4.2.0]oct-2-ene-2-ca...
Pharmaceutical Substances Syntheses, Patents, Applications - Part 113 potx
...
2-( methylthio )-
pyrrole
5-benzoyl- 2-( methyl- 6.6-dimethyl-5.7-dioxo-
1
-[ 2-( 4.6-dioxo-2.2-dimethyl-
thio)pyrrole
(11)
spiro[2.5]octone-
1,3-dioxon-5-yl)ethyl ]-2 -
4.8-dione (111)
(rnethy1thio )-5 -benzoylpyrrole ...
CN:
cis-
1
-acetyl- 4-[ 4-[ [ 2-( 2,4-dichloropheny1 )-2 -1
H-imidazol-1 -ylmethyl )- l,3-dioxolan- 4-
yl]methoxy]phenyl]p...