Pharmaceutical Substances Syntheses, Patents, Applications - Part 9 pot

... transcriptase inhibitor I RN: 13 647 0-7 8-5 MF: C,4H,uN60 MW: 286.34 1 CN: (1S,4R )-4 -[ 2-Amino- 6-( cyclopropylamino )-9 H-purin-9-yl ]-2 -cyclopentene-l-methanol succinate RN: 16 814 6-8 4-7 MF: Cl,HluN,O . ... 23.7 .19 91; appl. 22 .12 .19 89; GB-prior. 27.6 .19 88). d WO 9 924 4 31 (Glaxo; appl. 12 .1 1 .19 98; WO-prior. 12 .1 1 .19 97). alternative...

Ngày tải lên: 02/07/2014, 02:20

... levulinoyloxyacetate benzyl 1 2- ( 4-methoxyphenylhydrozano )- '=?' benzyl (5-meVloxy -2 - methyl-3-lndolyl- 4-chloro- benzoyl chloride benzyl [I -( 4-chlorobenzoyl )-5 -methoxy- 2- methyl-3-indolylocetoxy]acetate ... C,yH22N20S MW: 326 .46 EINECS: 23 6-6 6 1-9 LD,,: 517 mgkg (M, p.0.) CN: 1-[ l 0-[ 2- ( dimethylamino)propyl ]-1 0H-phenothiazin -2...

Ngày tải lên: 02/07/2014, 02:20

... 5 58 8- 1 6-9 MF: C,,H14C1N304S3 MW: 383 .90 EINECS: 22 6-9 9 4 -8 CN: 6-chloro-3,4-dihydro- 3-[ (2-propenylthio)methy1 ]-2 H- 1,2,4-benzothiadiazine-7-sulfonamide 1, l-dioxide 6-amino-4-chloro- chloroocetaldehyde ... hydrochloride CH3-CO-NH-NH2 , butanol - acetohydrazide 2-0 x 0-2 .3-dihydro-lH- 2-thioxo-2,3-dihydro- 7-chloro-5-phenyl-3H- 1.4-benzodiazepin...

Ngày tải lên: 02/07/2014, 02:20

... 3751 7-2 8-5 MF: C22H43NJ013 MW: 585.61 EINECS: 25 3-5 3 8-5 LD5,: 280 mgkg (M, i.v.); >6 glkg (M, p.0.) CN: (S)-O-3-amino-3-deoxy- ~-~ -glucopyranosyl-(1+6 )-0 -[ 6-amino-6-deoxy-a-u-glucopyranosyl-(l~4) ]- ... 298 499 (Res. Triangle Inst.; appl. 5.7. 199 1; USA-prior. 5.7. 199 1). WO 8 90 7 94 2 (US Bioscience; appl. 21.2. 198 9; USA-prior. 23.2. 198 8). US 5 167...

Ngày tải lên: 02/07/2014, 02:20

... 1-cyclohexyl-3-morpholinyl- ethyl-corbodiimide + N b VII H-Val-Tyr-Val-His-Pro-Phe-0-CH (VI) I-N ti2, ~d-C.CH~OH -m H H Z-Asn-Arg(N02)-Val-Tyr-Val-His-Pro-Phe-0-CH (W) 130 A Apalcillin ... Z-N 0 111 + HN,COOH \INYN/~0, H H Z -Asn-Arg(N0,)-OH (N) DMF, 1 -cyclahexyl- 3- morpholinylethyl-carbodiimide + I1 v Z-Val-Tyr-Val-His-Pro-Phe-0-CH (V) DMF, 1-cyc...

Ngày tải lên: 02/07/2014, 02:20

... 1,2,3.4-tetrahydro-6,7-dimethoxy- 2-isoquinolineprapionote [Ill) ethyl 1.3.4.6.7.1 1 b-hexohydm- N.N-diethyl-1.3.4.6.7,ll b-hexahydro-9.10. dimethoxy- 2-0 x 0-2 H- 9,lO-dimethaxy- 2-0 x 0-2 H- benzo[o]quinalizine- ... 6-chloro- 3-[ [(phenylmethyl)thio]methyl ]-2 H-1,2,4-benzothiadiazine-7-sulfonamide 1,l-dioxide 5-chloro-2.4-diomino- chloro- 7-ominonulfonyl-6-chloro-...

Ngày tải lên: 02/07/2014, 02:20

... 98 7-2 4-6 MF: C,H3,F06 MW: 434.50 EINECS: 21 3-5 7 8-6 CN: (1 1 ~,16~ )-2 1-( acetyloxy )-9 -fluoro-l1,17-dihydroxy-16-methylpregna-l,4-diene-3,20-dione 1. CH3-SO2-CI, pyridine 0 2. CH3-CO-NH-Br, ... anti-inflammatory, steroidal (BBP; TO- I 86) agent RN: 553 4-0 2-1 MF: C,,H,,F07 MW: 518.62 CN: (1 1 P, 16P )-9 -fluoro-1 I-hydroxy- 16-methyl- 1 7-( 1 -ox...

Ngày tải lên: 02/07/2014, 02:20

... RN: 3463 3-3 4-6 MF: C,,H,,F,O, MW: 292.33 CN: (R*,S* )-4 ,4&apos ;-( 1-ethyl-2-methyl-l,2-ethanediyl)bis[2-fluorophenol] 3-chloro- 2- trans-2.3-bis(3-fluora-4-methoxy- pentanone phenyl )-2 -pentene ... 20 0-3 9 9-3 CN: [3aS-(3aa,4~,6aa)]-hexahydro-2-oxo-1H-thieno[3,4-d]imidazole-4-pentanoic acid fumoric ocid mesa-2.3-dibromo- cis-1,3-dibenzyl- succinic ocid 2-axo...

Ngày tải lên: 02/07/2014, 02:20

... (? )-3 .4-dihydro- 4- hydroxy-2H-thieno- [3,2-el-1,2-thiozine 1 ,l -dioxide (111) hydride OH 1,3-dibromo- (? )-2 -( 3-bromopropyl )- propone 3,4-dihydro-4-hydroxy- 2H-thieno[3.2-el-1. 2- thiozine ... 1310 3-3 4-9 MF: C,,HN03 MW: 452.68 EINECS: 23 6-0 2 4-5 CN: (17~ )-1 7-[ (I-oxo-l0-undecenyl)oxy]androsta-l,4-dien-3-one boldenone RN: 84 6-4 8-0...

Ngày tải lên: 02/07/2014, 02:20

... ocetate. O°C XI1 - XI11 3-( brornoocetyl )- 5-chloro- 2- thiophenesulfonomide (XlIl) K2C03, DMSO XN + X b 4-hydroxy- 2-( 3-rnethoxy- propy1 )-2 H- thieno[3.2-el- 1,2-thiozine 1.1-dioxide (XV) ... oxolate Z-picaline 2-picoline ethyl 2-pyridyl- 1 -axide pyruvate 1'-oxide (In) 4-brornophenyl- hydrozine hydrochloride ethyl 5-brorno- 3- (2-pyridy1)ind...

Ngày tải lên: 02/07/2014, 02:20

... 143 1 .O6 CN: N-Acetyl- 3-( 2-naphthalenyl )-~ -alanyl-4-choro-~-phenyaanyl- 3-( 3-pyridinyl )-~ -alanyl-~-seryl- ~- tyrosyl- ~-( aminocarbonyl )-~ -ornithyl-~-leucyl-~-arginy ~-~ -prolyl-~-alaninamide ... 1765 0-9 8-5 MF: C5RH73N1302LS2 MW: 1352 .42 LD,,: 1012 mgkg (M, i.v.) CN: 5-oxo-~-prolyl-~-glutaminyl-~-a-asparty-O-sulfo-~-tyrosyl-~-threonylglycyl-~-tr...

Ngày tải lên: 02/07/2014, 02:20

... bronchodilator RN: 449 9-4 0-5 MF: C7H7N402. C5H,,N0 MW: 283.33 EINECS: 22 4-7 9 8-7 CN: 2-hydroxy-N,N,N-trimethylethanaminium, salt with 3,7-dihydro-l,3-dimethyl-IH-purine-2,6-dione (1:l) a-Chymotrypsin ... CN: (2R-trans )-2 -( 3,4-dihydroxyphenyl )-3 ,4-dihydro-2H-I-benzopyran-3,5,7-triol Cholestyramine C 453 Formulation(s): tabl. 250 mg, 500 mg Trade Name(s): D...

Ngày tải lên: 02/07/2014, 02:20

... 5986 5-1 3-3 MF: C,,Hll,N,,O,, MW: 1202.64 CN: [R-[R*,S *-( E)]]-cyclic(~-alanyl-~-alanyl-N-methyl-~-leucyl-N-methyl-~-leucyl-N-methyl-~-valyl- 3- hydroxy-N,4-dimethyl- ~-2 -amino-6-octenoyl-~-a-aminobutyryl-N-methylglycyl-N-methyl-~-leucyl- ~- ... hydrochloride methyl 5-cyclohexyl- 3-methyl- 5-0 x 0-2 - pentenoote (mixture with the 3-pentenoote: from methyl 4-me...

Ngày tải lên: 02/07/2014, 02:20

... RN: 2388 7-4 6-9 MF: Cz2H,,N3Os MW: 417.51 EINECS: 24 5-9 2 8-9 CN: 1-[ 2-oxo- 2-( l-pyrrolidinyl)ethyl ]-4 -[ l-oxo- 3-( 3,4,5-trimethoxyphcnyl)2-propenyl]pipera~ine maleate (1:l) RN: 2632 8-0 4-1 MF: ... 7569 6-0 2-5 MF: C,,H,,ClFN,O, MW: 357.77 LD,,,: 3.5 glkg (R, p.0.) 3.5 glkg (M, p.o) CN: (+ )-7 -Chloro- 5-( 2-fluorophenyl )-2 ,3-dihydro-...

Ngày tải lên: 02/07/2014, 02:20

... l 0-[ 3-( dimethylamino )-2 -methylpropyl ]-1 0H-phenothiazine-2-carbonitrile Z-chloropheno- thiozine P-cyanopheno- thiozine 1. NaNH2, xylene 2. cl&i:3 CH3 I 2. 1 -chloro-3-dimethyl- amino-2-methyl- Cyamemazine ... tonic RN: 63 3-4 7-6 MF: C,3H24N202 MW: 240.35 EINECS: 2 1 1-1 9 3-8 CN: N-[ 1-[ (dirnethylamino)carbonyI]propyl]-N-propyl-2-butenamid...

Ngày tải lên: 02/07/2014, 02:20