Pharmaceutical Substances Syntheses, Patents, Applications - Part 136 pdf

... hexofluorophosphote H3C-0 2. HCI H3C-0 H3C-0 0, 0, CH3 CH3 methyl N-benzoyl- 3.4-dimethoxy-L- phenylolanine. 1. HCI H3C-0 2. + 0=CH2 r 11 H3C-0 2. benzyl olcohol (S )-2 -amino- 3-( 3, 4- dimethoxypheny1 )- ... acetate Cl / N, \ \ / methyl 2-bromo- benzoate (-) -0 -chlorodiisopinocarnpheylborane. THF b methyl 2-[ 3-[ 3-[ (2E )-( 7-chloro- qui...

Ngày tải lên: 02/07/2014, 02:20

... (111) 4-pyridyl- molonoldehyde 1.2-dihydro- 2-0 x 0- 5-( 4-pyridyl). nicotinic acid 3-nitro- 5-( 4-pyridyl )- Z(1H)-pyridinone (IV) 120 A Anastrozole synthesis of ethyl N-(2,3-dichloro-6-aminobenzy1)glycinate: ... ester 2,3-dkhloro- 6-nitro- benzonitrile ethyl N-(2,3-dichloro- 6- diphenyl N-cyano- ethyl (2-cyonoimino-5, 6- orninobenzyi)glycinote irnidoc...

Ngày tải lên: 02/07/2014, 02:20

... 4-methyl- 2- nitrooniline 3-dimethylomino- 7- methyl-1,2-dihydro- 1,2,4-benzotriozine (I) NC, P43 HZ, Roney-Ni Y 4 b I CH, dimethyl- 3-dimethylomino-7methyl- cyonomide 1,2,4-benzotriozine ... 5 2-8 8-0 MF: Cl,H,,N,O, MW: 366.41 EINECS: 20 0-1 5 6-1 LD,,: 9300 pglkg (M, i.v.); 1320 mglkg (M, p.0.); 1902 mgkg (R, p.0.) CN: endo-(f )-3 -( 3-hydroxy-l-oxo-2-...

Ngày tải lên: 02/07/2014, 02:20

... ylthio)methyl ]-5 -thia-l-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid 7-orninocepholo- 4-mercopto- sporonic acid 1,Z.J-triozole 7(R)-omino- 3-[ (I ,2, 3- triozol-4-ylthio)methyl ]- 3-cephern-4-corboxylic ... RN: 5618 7-4 7-4 MF: C18H,5CI,N505S, MW: 548.45 CN: (6R-trans )-7 -[ [(3,5-dichloro-4-oxo-l(4H)-pyridinyl)acetyI]amino ]-3 -[ [(5-methyl-1,3,4-thiadiazol-...

Ngày tải lên: 02/07/2014, 02:20

... RN: 11 1 0-4 0-3 MF: C3,H3,N20s MW: 530.67 EINECS: 21 4-1 7 5-8 CN: (11~,16a )-2 1-( acetyloxy)-ll,17-dihydroxy-6,16-dimethyl-2'-phenyl-2'H-pregna-2,4,6-trieno[3, 2- clpyrazol-20-one Codeine ... 50 8-7 5-8 MF: C,H,,O,,, MW: 550.65 EINECS: 20 8-0 8 6-3 LD,,,: 1 mglkg (M, i.v.); >2 glkg (M, p.0.); 15.2 mg/kg (R, i.v.) CN: (3~,5~ )-3 -[ (6-deoxy-a...

Ngày tải lên: 02/07/2014, 02:20

... 2-mothyl-5,6,7, 8- 4-methylbenzyl- 2-methyl-1 -( 4-methyl- tctrahydroisoquino- mognesium chloride benzyl )-1 .2.5.6.7, 8- linium bromide hexohydroisoquinoline (+ )-2 -methyl- 1-( 4- methylbenzy1 )- ... 566 7-4 6-9 MF: C2,H2,N0,. H,PO, MW: 449.44 EINECS: 22 7-1 2 6-0 4-( 2-aminopropyl )- 1.2-dimethoxybenzene (I) 19 0-2 00 OC POCI, ___, n COOH...

Ngày tải lên: 02/07/2014, 02:20

... 5294 2-3 1-1 MF: C,9H28CINS0 MW: 377.92 CN: 2-[ 3-[ 4-( 3-chlorophenyl )-1 -piperazinyl]propyl ]-4 ,5-diethyl-2,4-dihydro-3H-1,2,4-triazol-3-one 4,5-diethyl- 1 -bromo- 3- 2-( 3-chloropropyl )- b 5-1 ... chlarobenzayl )- 5-ethylthiophene CH3COOH, pyridine - H\ 1- \ phosphorus - NH2 (I) 5-( 2-ch1orophenyl )- (11) 1.3-dihydro- 7...

Ngày tải lên: 02/07/2014, 02:20

... 4-( 3-formylpropyl )- carbonyl)propyl ]- hydride 1 -( trimethylsilyl )- 1H-imidazale imidozole (111) 4-( tert-butyl- 4-[ 4-[ 4-( tert-butyl- carbamoy1 )-1 - carbomoyl)-phenyll- 4- bromobenzene hydroxybutyl ]-1 -( trimethyl- ... [5R-[3(R*),5a,6a(R*)] ]-6 -( l-tlydroxyethyl )-7 -oxo- 3-( tetrahydro-2-furmyl )-4 -thia-l-azabicyclo[3.2.O ]...

Ngày tải lên: 02/07/2014, 02:20

... per- 2-nitro-5-fluoro- mongonote fluorotoluene benzoic acid HOOC ethyl isocyanate- 0 CH3 ocetote potossium tert-butylate N-methyl- 7-fluoro-4-methyl- glycine 3,4-dihydro-2H-1. 4- benzodiazepin-2,5(1H )- ... 8-fluoro-5,6-dihydro-5-methyl-6-oxo-4H-imidazo[l,5-a][1,4]be1uodiazepine-3-carhoxylic acid ethyl ester 1. Hz. Pd-C KMnO 2. COC12 F CH3 potassium F COOH 2....

Ngày tải lên: 02/07/2014, 02:20

... 2-[ [[ 1-( 4-chlorobenzoyl )-5 -methoxy-2-methyl-1H-indol-3-yl]acetyI]arnino ]-2 -deoxy-~-glucose indornetacin (9. v.) 1 -( 4-chlorobenzoyl )-2 - methyl-5-methoxyindol- 3-acetyl chloride (I) ... ethyl 2-( 2-methyl- 3.4.6-trifluorobenzayl )- 3-etho~yacr~late ethyl 2-( 2-methyl- 3.4.6-trifluorobenzoy1 )- 3-cyclopropylamino- acrylate (11) ethyl 1 -c...

Ngày tải lên: 02/07/2014, 02:20