Pharmaceutical Substances Syntheses, Patents, Applications - Part 11 pps
Pharmaceutical Substances Syntheses, Patents, Applications - Part 59 ppsx
...
RN: 101 1 6-2 2-0 MF: C2,Hz80z MW: 3 12.45 EINECS: 23 3-3 2 0-6
CN:
17-methyl-19-norpregna-4,9-diene-3,20-dione
3-rnethoxy-2 0-0 x 0-1 9-nor-
pregna-1,3.5(10).16-tetroene
(I)
(from estrone 3-methyl ...
RN: 60 4-5 1-3 MF:
C2,HZ7NO MW: 333.48 EINECS: 21 0-0 6 9-0
CN:
endo- 3-[ (l0,11-dihydro-5H-dibenzo[a,~cyclohepten-5-yl)oxy ]-8 -methyl-8-azabicyclo[3.2.l]oct...
Pharmaceutical Substances Syntheses, Patents, Applications - Part 5 pps
...
~-Alanyl-N-[(la,5a,6a )-3 -[ 6-carboxy- 8-( 2,4-difluoropheny )-3 -fluoro -5 , 8-dihydro -5 - oxo-l, 8-
naphthyridin-2-yl ]-3 -azabicyclo[3.1
.O]hex-6-yl]-L-alaninamide
monomethanesulfonate
base
RN: 14696 1-7 6-4 MF: C2,H2,F3N,0, MW: 55 8 .52
46
A
Alacepril ... 11 651 7; CP 11 651 7-2 7)
ATC: JOlMA
Use: antibacterial, prodrug
of
trovafloxacin
RN:
14696 1-7...
Pharmaceutical Substances Syntheses, Patents, Applications - Part 10 pps
...
2-amino- 7-(
I-methylethyl )-5 -0 x0-SH-[I
~henzopyrano[2,3-b]pyr1dine-3-carhc~xyl~c
ac~d
2-hydroxy-5-isopropyl- dimelhyl- 6-isopropy- 4-0 x 0-
acetophenone formornide
4H-1
-benzopyran- 3-
corboxaldehyde ...
DMF
1
-
H3C
hydroxylomine
CN
morpholinc
.
dimethyl-
CHO
CH3
*
formornnde
.
CH3
0
6-ixopropyl-4-oro- 2-amino-6-isopropyl-
4H-
I-
benropyron- 4...
Pharmaceutical Substances Syntheses, Patents, Applications - Part 11 pps
...
RN: 7095 8-8 6-0 MF: Cl,H,N,05S
.
HCI MW: 416.93
Guoiacol 1,2-dibromo-
(2-rnethoxy- ethane
phenol)
3-amino-4-methyl-
acetaphenone
5-acetyl-2-methyl-
benzenesulfanornide
5-[ [N-[ 2-( 2-rnethoxyphenoxy)ethyl ]- ... EINECS: 24 8-0 0 3-8
LD,,:
>25 gkg (M, p.0.);
>15
gkg
(R, p.0.)
CN:
[2S-[2a,5a,6~(S*)] ]-6 -[ [amino(4-hydroxyphenyl)acetyl]amino ]-3 ,3-...
Pharmaceutical Substances Syntheses, Patents, Applications - Part 20 ppsx
...
2-0 x 0-2 .5-dihydro- chloride (2.5-dihydro-50x 0-
furon
3-furyl)ocetophenone
d'
I,
0
boranote
4&apos ;-( 2.5-dihydro- 5-0 x 0-
2-acetyl- 5-( 2.5-dihydro-
5-( 2.5-dihydro-50x 0-
3-furyl )-2 &apos ;-( 2-oxopropaxy )- ... vasodilator
RN: 344 7-9 5-8 MF:
C,,H1807 MW: 358.35 EINECS: 22 2-3 6 7-8
LD,,: 520 mglkg (M, p.0.)
CN: butanedioic a...
Pharmaceutical Substances Syntheses, Patents, Applications - Part 31 pps
...
RN:
6455 2-1 7-6
MF:
C,,H,$NO,
MW:
31
1.40
CN:
(~ )-1 -[ 2-[ 3-[ (1,1-dimethylethyl)amino ]-2 -hydroxypropoxy ]-5 -fluorophenyl]-I-butanone
phenol chloride butyrophenone
tert-butyl-
amine
Butofilolol ...
21 mgkg
(R,
i.v.)
CN:
[3(S)-endo ]-8 -[ (4-butoxyphenyl)methyl ]-3 -( 3-hydroxy-1-oxo-2-phenylpropoxy )-8 -methyl- 8-
azoniabicyclo[3.2. lloctane...
Pharmaceutical Substances Syntheses, Patents, Applications - Part 32 pps
...
RN: 5816 6-8 3-9 MF: C,,H,,N,O,
MW:
357.41
CN:
3,7-dihydro- 7-[ 2-[ (2-hydroxy-l-methyl-2-phenylethyl)amino]ethyl ]-1 ,3-dimethy-1
H-purine-2,6-dione
[R-(R*,S*)]-cafedrine
RN: 7839 6-3 4-6 MF: C,,H,,N,O, ... 8140 9-9 0-7 MF: C,,H,,N,O, MW: 451.62
CN:
(8~)-N-[ 3-( Dirnethylamino)propyl]-N-[(ethylamino)carbonyl ]-6 -( 2-propenyl)ergoline-8-carboxamide
1.
K2C03...
Pharmaceutical Substances Syntheses, Patents, Applications - Part 51 ppsx
... 424.99 EINECS: 24 2-2 0 9-1
LDso: 2618 mgkg (R, s.c.)
CN:
(2s-trans)-methyl
7-chloro-6,7,8-trideoxy- 6-[ [(I
-methyl-4-propyl-2-pyrrolidinyl)carbonyl]amino]-l-thio-
L-threo-a-D-gulucto-octopyranoside ... mglkg (R, p.0.)
CN: 7-chloro-1 -methyl-5-phenyl- 1
H-
1.5-benzodiazepine-2,4(3H,SH)-dione
1
-3 -dichloro-
benzene
CI
nNo2
6
5-chloro- 2-
nitrodiphenyl-
arnine
(I...
Pharmaceutical Substances Syntheses, Patents, Applications - Part 52 ppsx
...
RN: 192 6-4 9-4 MF: C17H,,C12N205S MW: 433.3 1 EINECS: 21 7-6 5 7-6
CN:
[2S-(2a,5a,6~) ]-6 -[ [(3,4-dichlorophenyl)methoxyacetyl]amino ]-3 ,3-dimethyl-7-oxo-4-thia- 1-
azabicyclo[3.2.0]heptane-2-carboxylic ...
482 8-2 7-7 MF: C2,H2,C1FO4 MW: 41 0.9 1 EINECS: 22 5-4 0 6-7
CN:
(6a,l
I
P,l6a )-9 -chloro-6-fluoro-
1
I
,2 1 -dihydroxy-
16-methylpregna-1,4-die...
Pharmaceutical Substances Syntheses, Patents, Applications - Part 150 pps
... Orlipastat; Ro- 1 8-0 647) Use: antiobesity, pancreatic lipase inhibitor
RN:
9682 9-5 8-2 MF: C2,Hs3NOs MW: 495.75
CN:
N-Formyl-t-leucine
[2S-[2a(R*),3.beta.]]-l-[[3-hexyl-4-oxo-2-oxetanyl]methyl]dodecyl ...
' 1-
OHC-
2.
pyridinium
(CH2)
, 0-
CH3
dichrornote
3(R)-benzyloxy-
tetrodeconol (XVII)
Orgotein
0
1493
3',5'-dirnethoxyaceto-
2-brorno-Y.5&a...
Pharmaceutical Substances Syntheses, Patents, Applications - Part 61 pps
...
RN:
3902 6-3 9-6 MF: C,H,,FO, MW: 654.90 EINECS: 25 4-2 5 4-4
CN: [ll
~,16a,2 1-( Z,Z) ]-9 -fluoro-l1,17-dihydroxy-
16-methyl-2l-[(l-oxo-9,12-octadecadienyl)oxy]-pregna-
1,4-diene-3,20-dione
dexamethasane ... 20 6-2 3 2-0
CN:
(1
1
P,
l6a)-Y-fluoro-l l ,
17-dihydroxy-
16-methy 1-2 1-( phosphonooxy)pregna-1,4-diene-3,20-dione
disodium
salt
RN:
239 2-3 9-...
Pharmaceutical Substances Syntheses, Patents, Applications - Part 64 pps
...
RN: 31 1 6-7 6-5 MF: C,9Hl,CIZN30sS MW: 470.33 EINECS: 221 -4 8 8-3
CN:
[2S-(2a,5a,6~) ]-6 -[ [[ 3-( 2,6-dichlorophenyl )-5 -methyl-4-isoxazolyl]carbonyl]amino ]-3 ,3-dimethyl- 7-
oxo-4-thia-l-azabicyclo[3.2.0]heptane-2-carboxylic ...
1
1 P,16a )-6 ,9-difluoro- 1 1-hydroxy-
16-methyl-2 1-[ (1-oxopentyl)oxy]pregna-1,4-diene-3,20-dione
diflucortolone
RN: 260 7...
Pharmaceutical Substances Syntheses, Patents, Applications - Part 68 ppsx
... 52 0-2 7-4
MF:
C2,H,,OI5 MW: 608.55 EINECS: 20 8-2 8 9-7
CN:
7-[ [6-O-(6-deoxy-a-~-mannopyranosyl )-~ -~ -glucopyranosyl]oxy ]-5 -hydroxy- 2-( 3-hydroxy- 4-
methoxypheny1 )-4 H-1 -benzopyran-4-one
680 ...
(Jodopyracet)
Use: X-ray contrast medium
RN: 101 -2 9-1 MF: C7H512N03 MW: 404.93 EINECS: 20 2-9 3 2-5
CN:
3,5-diiodo- 4-0 x0-l(4H)-pyridineacetic...
Pharmaceutical Substances Syntheses, Patents, Applications - Part 75 ppsx
...
[2S-[2a,Sa,6P(S*)] ]-6 -[ (amino-
1,4-cyclohexadien- 1
-ylacetyl)amino ]-3 ,3-dimethyl-7-oxo-4-thia-
1
-
azabicyclo[3.2.0]heptane-2-carboxylic
acid
monosodium salt
RN: 3473 5-4 0-5 MF: C,,H,N,NaO,S MW: 373.41
750 ... yN-"tw2
+
H2N*NH2
/
0
methyl 4-benzyloxy- ethylene-
N-(2-arninoethy1 )-4 -benzyloxy-
phenylacetate
diamine phenylacetarnide
(1)
1.2-epoxy-...
Pharmaceutical Substances Syntheses, Patents, Applications - Part 76 pps
...
p.0.)
CN:
4-methoxy- 2-( 5-methoxy-3-methyl-lH-pyrazol-l-yl )-6 -methylpyrimidine
,
I
hydmzine
OH
CI
0,
CH3
hydrote
6-methyl- 2,4-dichloro- 2-chloro- 4-
uracil
6-methyl-
methoxy- 6-
pyrimidine ...
(8S-cis)-l 0-[ (3-amino-2,3,6-trideo~y-a-~-alnbino-hexopyranosyl)oxy ]-7 ,8,9,1O-tetrahydro-6,8,1 1-
trihydroxy- 8-( hydroxyacety1 )-
I
methoxy-5,12-naphtha...